TargetNet


P00760

Cationic trypsin


Function

Not available.


Database Links

Database Links
UniProt P00760
PDB 1AQ7, 1AUJ, 1AZ8, 1BJU, 1BJV, 1BTP, 1BTW, 1BTX, 1BTY, 1BTZ, 1C1N, 1C1O, 1C1P, 1C1Q, 1C1R, 1C1S, 1C1T, 1C2D, 1C2E, 1C2F, 1C2G, 1C2H, 1C2I, 1C2J, 1C2K, 1C2L, 1C2M, 1C5P, 1C5Q, 1C5R, 1C5S, 1C5T, 1C5U, 1C5V, 1C9T, 1CE5, 1CU7, 1CU8, 1CU9, 1D6R, 1EB2, 1EJM, 1EZX, 1F0T, 1F0U, 1F2S, 1G36, 1G3B, 1G3C, 1G3D, 1G3E, 1G9I, 1GBT, 1GHZ, 1GI0, 1GI1, 1GI2, 1GI3, 1GI4, 1GI5, 1GI6, 1GJ6, 1HJ9, 1J8A, 1JIR, 1JRS, 1JRT, 1K1I, 1K1J, 1K1L, 1K1M, 1K1N, 1K1O, 1K1P, 1LQE, 1MAX, 1MAY, 1MTS, 1MTU, 1MTV, 1MTW, 1N6X, 1N6Y, 1NC6, 1NTP, 1O2H, 1O2I, 1O2J, 1O2K, 1O2L, 1O2M, 1O2N, 1O2O, 1O2P, 1O2Q, 1O2R, 1O2S, 1O2T, 1O2U, 1O2V, 1O2W, 1O2X, 1O2Y, 1O2Z, 1O30, 1O31, 1O32, 1O33, 1O34, 1O35, 1O36, 1O37, 1O38, 1O39, 1O3A, 1O3B, 1O3C, 1O3D, 1O3E, 1O3F, 1O3G, 1O3H, 1O3I, 1O3J, 1O3K, 1O3L, 1O3M, 1O3N, 1O3O, 1OPH, 1OX1, 1OYQ, 1P2I, 1P2J, 1P2K, 1PPC, 1PPE, 1PPH, 1QA0, 1QB1, 1QB6, 1QB9, 1QBN, 1QBO, 1QCP, 1QL7, 1QL8, 1RXP, 1S0Q, 1S0R, 1SBW, 1SFI, 1SMF, 1TAB, 1TAW, 1TGB, 1TGC, 1TGN, 1TGS, 1TGT, 1TIO, 1TLD, 1TNG, 1TNH, 1TNI, 1TNJ, 1TNK, 1TNL, 1TPA, 1TPO, 1TPP, 1TPS, 1TX7, 1TX8, 1TYN, 1UTN, 1UTO, 1UTP, 1UTQ, 1V2J, 1V2K, 1V2L, 1V2M, 1V2N, 1V2O, 1V2P, 1V2Q, 1V2R, 1V2S, 1V2T, 1V2U, 1V2V, 1V2W, 1XUF, 1XUG, 1XUH, 1XUI, 1XUJ, 1XUK, 1Y3U, 1Y3V, 1Y3W, 1Y3X, 1Y3Y, 1Y59, 1Y5A, 1Y5B, 1Y5U, 1YP9, 1YYY, 1ZR0, 1ZZZ, 2A7H, 2AGE, 2AGG, 2AGI, 2AH4, 2AYW, 2BLV, 2BLW, 2BTC, 2BY5, 2BY6, 2BY7, 2BY8, 2BY9, 2BYA, 2BZA, 2CMY, 2D8W, 2F3C, 2FI3, 2FI4, 2FI5, 2FTL, 2FTM, 2FX4, 2FX6, 2G55, 2G5N, 2G5V, 2G81, 2G8T, 2ILN, 2J9N, 2O9Q, 2OTV, 2OXS, 2PLX, 2PTC, 2PTN, 2QN5, 2QYI, 2TGA, 2TGD, 2TGP, 2TGT, 2TIO, 2TLD, 2TPI, 2UUY, 2XTT, 2ZDK, 2ZDL, 2ZDM, 2ZDN, 2ZFS, 2ZFT, 2ZHD, 2ZQ1, 2ZQ2, 3A7T, 3A7V, 3A7W, 3A7X, 3A7Y, 3A7Z, 3A80, 3A81, 3A82, 3A83, 3A84, 3A85, 3A86, 3A87, 3A88, 3A89, 3A8A, 3A8B, 3A8C, 3A8D, 3AAS, 3AAU, 3AAV, 3ATI, 3ATK, 3ATL, 3ATM, 3BTD, 3BTE, 3BTF, 3BTG, 3BTH, 3BTK, 3BTM, 3BTQ, 3BTT, 3BTW, 3D65, 3E8L, 3GY2, 3GY3, 3GY4, 3GY5, 3GY6, 3GY7, 3GY8, 3I29, 3ITI, 3LJJ, 3LJO, 3M35, 3M7Q, 3MFJ, 3MI4, 3NK8, 3NKK, 3OTJ, 3PLB, 3PLK, 3PLP, 3PM3, 3PMJ, 3PTB, 3PTN, 3PWB, 3PWC, 3PYH, 3Q00, 3QK1, 3RDZ, 3RU4, 3RXA, 3RXB, 3RXC, 3RXD, 3RXE, 3RXF, 3RXG, 3RXH, 3RXI, 3RXJ, 3RXK, 3RXL, 3RXM, 3RXO, 3RXP, 3RXQ, 3RXR, 3RXS, 3RXT, 3RXU, 3RXV, 3T25, 3T26, 3T27, 3T28, 3T29, 3TPI, 3UNQ, 3UNR, 3UNS, 3UOP, 3UPE, 3UQO, 3UQV, 3UUZ, 3UWI, 3UY9, 3V0X, 3V12, 3V13, 3VEQ, 3VPK, 4AB8, 4AB9, 4ABA, 4ABB, 4ABD, 4ABE, 4ABF, 4ABG, 4ABH, 4ABI, 4ABJ, 4AOQ, 4AOR, 4B1T, 4B2A, 4B2B, 4B2C, 4GUX, 4HGC, 4I8G, 4I8H, 4I8J, 4I8K, 4I8L, 4J2Y, 4TPI, 5PTP
BioGrid Not available
BindingDB P00760
DrugBank DB01093
Guide to PHARMACOLOGY Not available
PharmGKB Not available
KEGG bta:615026, bta:780933
BioCyc Not available
Entrez Gene (GeneID) 615026, 780933

Chemical Space of the Positive Compounds


Model Performance Metrics

Metric Mean Value Standard Deviation
AUC 0.9376 0.0034
Accuracy 0.8851 0.0034
Sensitivity 0.9198 0.0066
Specificity 0.8452 0.0053
BEDROC 0.976 0.0115
MCC Threshold 0.516 N/A
MCC 0.7746 N/A
F-score Threshold 0.516 N/A
F-score 0.8974 N/A

Downloads

R Model Object

Random Forest model object (.RData)

Download RData

Positive Set

SMILES string + affinity value (.tsv)

Download TSV


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Page generated on: 2014-04-29 14:39:17